Effects of 4-aminopyridine on attention and executive functions of patients with multiple sclerosis: Randomized, double-blind, placebo-controlled clinical trial. Preliminary report


Por: Arreola-Mora C., Silva-Pereyra J., Fernández T., Paredes-Cruz M., Bertado-Cortés B., Grijalva I.

Publicada: 1 feb 2019
Resumen:
Background: A high percentage of patients with multiple sclerosis present cognitive alterations. Because 4-aminopyridine improves nerve conduction and efficient synaptic connection could improve cognitive dysfunction. Objective: To evaluate the efficacy on cognitive performance and safety of 4-aminopyridine administered to patients with relapsing-remitting multiple sclerosis. Methods: A randomized, double-blind, placebo controlled clinical trial was conducted in patients with relapsing-remitting multiple sclerosis diagnosis according to the McDonald criteria. At the beginning and at the end of the treatment different tests were used to assess cognitive performance. Subsequently, patients were randomized 1:1 to receive treatment or placebo. A bootstrap-t test was proposed to test the effectiveness of cognitive performance, considering a p-value < 0.05 as statistically significant. Results: Twenty-four patients were recruited of which 21 completed the trial, 11 with 4-aminopyridine and 10 with placebo treatment. No significant differences between groups in the initial assessments were observed. In terms of efficacy, the experimental group achieved significantly higher scores in attention span, verbal fluency, planning and graphics and constructive motion. Conclusions: 4-aminopyridine proved to be an effective treatment on cognitive aspects in patients with relapsing-remitting multiple sclerosis. Drug doses were shown to be safe with mild to moderate adverse events.

Filiaciones:
Arreola-Mora C.:
 Laboratorio de Neurometría, Proyecto de Neurociencias, Facultad de Estudios Superiores Iztacala, Universidad Nacional Autónoma de México, Mexico City, Mexico

 Unidad de Investigación Médica de Enfermedades Neurológicas, Unidad Médica de Alta Especialidad, Hospital de Especialidades, Centro Médico Nacional Siglo XXI, Instituto Mexicano del Seguro Social, Cuauhtémoc 330. Col. Doctores. C. P, Mexico City, 06720, Mexico

 Univ Nacl Autonoma Mexico, Fac Estudios Super Iztacala, Lab Neurometria, Proyecto Neurociencias, Mexico City, DF, Mexico

 Hosp Especialidades Ctr Med La Raza, Ctr Med Nacl Siglo XXI, Inst Mexicano Seguro Social, Unidad Med Alta Especialidad,Unidad Invest Med En, Cuauhtemoc 330 Col Doctores, Mexico City 06720, DF, Mexico

Silva-Pereyra J.:
 Laboratorio de Neurometría, Proyecto de Neurociencias, Facultad de Estudios Superiores Iztacala, Universidad Nacional Autónoma de México, Mexico City, Mexico

 Univ Nacl Autonoma Mexico, Fac Estudios Super Iztacala, Lab Neurometria, Proyecto Neurociencias, Mexico City, DF, Mexico

Fernández T.:
 Departamento de Neurobiología Conductual y Cognitiva, Instituto de Neurobiología, Universidad Nacional Autónoma de México, Campus UNAM-UAQ, Juriquilla, Queretaro, Mexico

 Univ Nacl Autonoma Mexico, Inst Neurobiol, Dept Neurobiol Conductual & Cognit, Campus UNAM UAQ, Juriquilla, Queretaro, Mexico

Paredes-Cruz M.:
 Unidad de Investigación Médica de Enfermedades Neurológicas, Unidad Médica de Alta Especialidad, Hospital de Especialidades, Centro Médico Nacional Siglo XXI, Instituto Mexicano del Seguro Social, Cuauhtémoc 330. Col. Doctores. C. P, Mexico City, 06720, Mexico

 Hosp Especialidades Ctr Med La Raza, Ctr Med Nacl Siglo XXI, Inst Mexicano Seguro Social, Unidad Med Alta Especialidad,Unidad Invest Med En, Cuauhtemoc 330 Col Doctores, Mexico City 06720, DF, Mexico

Bertado-Cortés B.:
 Departamento de Neurología, Unidad Médica de Alta Especialidad, Hospital de Especialidades, Centro Médico Nacional Siglo XXI, Instituto Mexicano del Seguro Social, Mexico City, Mexico

 Hosp Especialidades Ctr Med La Raza, Ctr Med Nacl Siglo XXI, Inst Mexicano Seguro Social, Dept Neurol,Unidad Med Alta Especialidad, Mexico City, DF, Mexico

Grijalva I.:
 Unidad de Investigación Médica de Enfermedades Neurológicas, Unidad Médica de Alta Especialidad, Hospital de Especialidades, Centro Médico Nacional Siglo XXI, Instituto Mexicano del Seguro Social, Cuauhtémoc 330. Col. Doctores. C. P, Mexico City, 06720, Mexico

 Hosp Especialidades Ctr Med La Raza, Ctr Med Nacl Siglo XXI, Inst Mexicano Seguro Social, Unidad Med Alta Especialidad,Unidad Invest Med En, Cuauhtemoc 330 Col Doctores, Mexico City 06720, DF, Mexico
ISSN: 22110348
Editorial
Elsevier, THE BOULEVARD, LANGFORD LANE, KIDLINGTON, OXFORD OX5 1GB, OXON, ENGLAND, Reino Unido
Tipo de documento: Article
Volumen: 28 Número:
Páginas: 117-124
WOS Id: 000459833100023
ID de PubMed: 30593980

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